Pregabalin

Salts []
Pregabalin hydrochloride
Sodium pregabalin

Molecular structure via molpic
Conformer structure via 3Dmol.js
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Molecular formula	C8H17NO2[1]
Molecular mass	159.23 g/mol[1]
Appearance	White to off-white crystalline solid[1]
Predicted LogP	-1.6[1]
Melting point	186-188 °C[1]
Solubility	Freely soluble[1]
Chirality	absolute[2]

Identifiers []
IUPAC name	(3S)-3-(aminomethyl)-5-methylhexanoic acid[1]
SMILES	CC(C)C[C@@H](CC(=O)O)CN[1]
InChI	InChI=1S/C8H17NO2/c1-6(2)3-7(5-9)4-8(10)11/h6-7H,3-5,9H2,1-2H3,(H,10,11)/t7-/m0/s1[1]
InChIKey	AYXYPKUFHZROOJ-ZETCQYMHSA-N[1]

Dosing
Elimination half-life	4.5 – 7 hours[4] (mean 6.3 hours)[5]
Duration of action	8 – 12 hours [6]

Pregabalin

Pregabalin (also known as (S)-3-(Aminomethyl)-5-methylhexanoic acid, 3-isobutyl GABA, (S)-Pregabalin, Pregabalina, Pregabaline, Vronogabic, Pregabalin mylan, Pregabalin sandoz, Pregabalin zentiva or Pregabalin sandoz gmbh) is a substance of the gabapentinoid class.

Chemistry

Pregabalin is typically found in the form of its hydrochloride and sodium salts.

Stereochemistry

Pregabalin is a absolute mixture

Subjective effects

Experience reports

There are currently 25+ experience reports involving pregabalin on OpenErowid: []

• "Observations Over 4 Years of Usage"
• "Amazing Time Slip"
• "My Hellish Withdrawal"
• "I Wish I Hadn't Redosed"
• "Painless Time and Zoned Out"
• "My Social Anxiety Has Been Obliterated"
• "Long-Term Use and High Dosages"
• "Closed Eye Visuals Similar to Lucid Dreaming"
• "Wishing It Never Ended"
• "All in Around 5 Years"
• "On a Dose for a Traumatic Brain Injury"
• "A Very Romantic Night With My Wife"
• "Gentle and Smooth"
• "Ghost In My Kitchen"
• "Cannabis Type Buzz"
• "The Journey Into Acceptance"
• "Mildly Dissociative"
• "Personal Effects Summary"
• "I Can Alter the Scene-Flow"
• "Cutting-Edge Pharmacology a Double-Edged Swor"
• "Effects Peaked Around the Two Hour Mark"
• "Body Warmth and Pleasantness of Mind"
• "A Little Too Much"
• "Zero Recreational Benefits"
• "Maybe Mania"

Legal status

• Australia: Pregabalin is a S4 substance.^[3]
• Brazil: Pregabalin is a C1 substance.
• Canada: Pregabalin is a prescription only substance.
• New Zealand: Pregabalin is a prescription only substance.
• United Kingdom: Pregabalin is a prescription only substance.
• United States: Pregabalin is a Schedule V substance.
• European Union: Pregabalin is a prescription only substance.

See also

• Calcium Channel Blocker
• Substituted gabapentinoids
• Anodyne

External links

• Pregabalin (Wikipedia)
• Pregabalin (Wikidata)
• Pregabalin (DrugBank)
• Pregabalin (PubChem)
• Pregabalin (ChEMBL)
• Pregabalin (ChEBI)
• Pregabalin (Probes & Drugs)
• Pregabalin (Common Chemistry)
• Pregabalin (HMDB)
• Pregabalin (KEGG)
• Pregabalin (UNII)
• Pregabalin (EPA DSSTox)

References