Anodyne| EC | |
|---|---|
| Molecular structure via molpic based on CDK |
| Conformer [] | |
|---|---|
| Conformer structure via JSmol | |
| Physical properties [] | |
|---|---|
| Molecular mass | 396.6 g/mol [1] |
| Predicted LogP | 7.1 [1] |
| Structural Identifiers [] | |
|---|---|
| Molecular formula | C26H36O3 [1] |
| IUPAC name | [(8R,9S,13S,14S,17S)-3-hydroxy-13-methyl-6,7,8,9,11,12,14,15,16,17-decahydrocyclopenta[a]phenanthren-17-yl] 3-cyclopentylpropanoate [1] |
| SMILES | C[C@]12CC[C@H]3[C@H]([C@@H]1CC[C@@H]2OC(=O)CCC4CCCC4)CCC5=C3C=CC(=C5)O [1] |
| InChI | InChI=1S/C26H36O3/c1-26-15-14-21-20-10-8-19(27)16-18(20)7-9-22(21)23(26)11-12-24(26)29-25(28)13-6-17-4-2-3-5-17/h8,10,16-17,21-24,27H,2-7,9,11-15H2,1H3/t21-,22-,23+,24+,26+/m1/s1 [1] |
| InChIKey | UOACKFBJUYNSLK-XRKIENNPSA-N [1] |
| Dosing [] | |
|---|---|
| Elimination half-life | Intramuscular injection (aqueous suspension): 8 – 10 days[3] |
| Duration of action | Intramuscular injection (oil solution|oil): 5 mg ≈ 11 – 14 days[4]Intramuscular injection (aqueous suspension): 5 mg ≈ 14 – 24 days |
Estradiol cypionate
(Redirected from estradiol cypionate)
Estradiol cypionate (also known as Depoestradiol, Depofemin, Depo-Estradiol, Depoestra, Estradep, Estrapo, Estro-Depo, Dep-Estro, Femogen CYP or β-Estradiol 17-cypionate)
Chemistry
Stereochemistry []
Estradiol cypionate is a absolute mixture
| Anodyne Usernotes [] | |
|---|---|
| 0xea / Estradiol cypionate via | Prodrug Ester of Estradiol; crashes when injected weekly |
See also []
External links []
- Estradiol cypionate (Wikipedia)
- Estradiol cypionate (Wikidata)
- Estradiol cypionate (DrugBank)
- Estradiol cypionate (PubChem)
- Estradiol cypionate (ChEMBL)
- Estradiol cypionate (ChEBI)
- Estradiol cypionate (Common Chemistry)
- Estradiol cypionate (KEGG)
- Estradiol cypionate (UNII)
- Estradiol cypionate (EPA DSSTox)
References []
National Center for Biotechnology Information. PubChem Compound Summary for CID 9403, Estradiol cypionate. Accessed July 7, 2025. https://pubchem.ncbi.nlm.nih.gov/compound/9403
U.S. Food and Drug Administration; National Center for Advancing Translational Sciences. Estradiol cypionate. UNII: 7E1DV054LO. Global Substance Registration System. Accessed July 7, 2025. https://gsrs.ncats.nih.gov/ginas/app/beta/substances/7E1DV054LO
Thurman A, Kimble T, Hall P, Schwartz JL, Archer DF. Medroxyprogesterone acetate and estradiol cypionate injectable suspension (Cyclofem) monthly contraceptive injection: steady-state pharmacokinetics. Contraception. June 1, 2013; 87(6):738–43.
Oriowo MA, Landgren BM, Stenström B, Diczfalusy E. A comparison of the pharmacokinetic properties of three estradiol esters. Contraception. April 1, 1980; 21(4):415–24.